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Search Results for " histamine receptor "

20

Compounds

Cat No. Product Name Synonyms Targets
T38634 Histamine H4 receptor antagonist-1 Histamine H4 receptor antagonist-1
Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.
T0965 Histamine Ergamine 5-HT Receptor , Endogenous Metabolite , Histamine Receptor
Histamine (Ergamine) is an amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial smooth muscle, a vasodilator, and also a centrally acting ne...
T10680 Carebastine Histamine Receptor
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
T9717 Chlorcyclizine HCV Protease , Histamine Receptor
CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.
T22842 HTMT dimaleate Histamine Trifluoromethyl Toluidide Dimaleate Histamine Receptor
HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.
T22724 Dimaprit dihydrochloride NOS , NO Synthase , Histamine Receptor
Dimaprit dihydrochloride is a selective histamine H2 receptor agonist. Dimaprit dihydrochloride also inhibits nNOS with an IC50 of 49 μM. It can stimulate gastric acid secretion.
T9353 OXOMEMAZINE AChR , Histamine Receptor
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M1 receptors, showing high (Ki=84 nM, M1 receptors) and low ...
T7477 Antazoline Others
Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.
T8439 Clobenpropit dihydrobromide Apoptosis , Histamine Receptor
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
T5829 H4 Receptor antagonist 1 Histamine Receptor
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
T4563 Thonzylamine neohetramine Histamine Receptor
Thonzylamine (neohetramine) is an antihistamine and anticholinergic drug. It is available as combination products with Clofedanol or Phenylephrine for temporary relief of symptoms of common cold, hay fever (allergic rhin...
T19680 Zotepine Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM, 3.3 nM, 7.3 nM, and 8 nM, respectively. Zotepine is a second...
T7085 Mebhydrolin Mebhydroline Histamine Receptor
Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.
T4250 Bilastine Bilaxten Histamine Receptor
Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of action.
T11723L JNJ-39758979 Histamine Receptor
JNJ-39758979 is a selective and high-affinity histamine H4 receptor antagonist (Kis: 12.5, 5.3, and 25 nM for human, mouse, and monkey histamine H4 receptor, respectively). JNJ-39758979 functionally antagonizes histamine...
T36949 Niaprazine 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for sleep disorder research[1][2]. Niaprazine exhibits a low aff...
T20712 Conessine Conessinum,Wrightine,Roquessine,Neriine,Konessin Histamine Receptor
Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.
T7564 Chlorphenoxamine Contristamine Histamine Receptor
Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
T1278 Astemizole Laridal,Histaminos,Paralergin Potassium Channel , Histamine Receptor
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to re...
T12489 Pimethixene Calmixen,Pimetixene Dopamine Receptor , 5-HT Receptor , AChR , Histamine Receptor
Pimethixene (Calmixen) is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 ...

Compounds

Histamine H4 receptor antagonist-1
T38634
Synonym: Histamine H4 receptor antagonist-1
Target:
Histamine
T0965
Synonym: Ergamine
Target: 5-HT Receptor, Endogenous Metabolite, Histamine Receptor
Carebastine
T10680
Synonym:
Target: Histamine Receptor
Chlorcyclizine
T9717
Synonym:
Target: HCV Protease, Histamine Receptor
HTMT dimaleate
T22842
Synonym: Histamine Trifluoromethyl Toluidide Dimaleate
Target: Histamine Receptor
Dimaprit dihydrochloride
T22724
Synonym:
Target: NOS, NO Synthase, Histamine Receptor
OXOMEMAZINE
T9353
Synonym:
Target: AChR, Histamine Receptor
Antazoline
T7477
Synonym:
Target: Others
Clobenpropit dihydrobromide
T8439
Synonym:
Target: Apoptosis, Histamine Receptor
H4 Receptor antagonist 1
T5829
Synonym:
Target: Histamine Receptor
Thonzylamine
T4563
Synonym: neohetramine
Target: Histamine Receptor
Zotepine
T19680
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Mebhydrolin
T7085
Synonym: Mebhydroline
Target: Histamine Receptor
Bilastine
T4250
Synonym: Bilaxten
Target: Histamine Receptor
JNJ-39758979
T11723L
Synonym:
Target: Histamine Receptor
Niaprazine
T36949
Synonym:
Target: 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Conessine
T20712
Synonym: Conessinum,Wrightine,Roquessine,Neriine,Konessin
Target: Histamine Receptor
Chlorphenoxamine
T7564
Synonym: Contristamine
Target: Histamine Receptor
Astemizole
T1278
Synonym: Laridal,Histaminos,Paralergin
Target: Potassium Channel, Histamine Receptor
Pimethixene
T12489
Synonym: Calmixen,Pimetixene
Target: Dopamine Receptor, 5-HT Receptor, AChR, Histamine Receptor
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TargetMol